WORKSHOP II - A DECADE OF STRUCTURE-BASED DRUG DESIGN

Lectures

Regency Ballroom C (RC)

Saturday, July 19




08:30 - 08:35 AM
Opening Remarks. S. Abdel-Meguid, Presiding.

08:35 - 09:20 AM
Wim Hol. Invited Lecture.
Structure- Based Drug Design - A Meeting Place of Angstroms, Kilocals, Insight, Serendipity and Creativity.

09:20 - 10:05 AM
Christine Humblet. Invited Lecture.
Computer-Based Approaches in Structure- Based Design.

10:05 - 10:30 AM
Coffee Break.

10:30 - 11:15 AM
Michael Varney. Invited Lecture.
Protein Structure- Based Molecular Design as a Tool in Drug Discovery. What We Have Learned in the Last 10 Years.

11:15 - 12:00 AM
Stephen Fesik. Invited Lecture.
SAR by NMR: A Method for Discovering High Affinity Ligands.

01:30 - 02:00 PM WII01
(E167)
Ravi G. Kurumbail. Invited Lecture.
Structure- Based Drug Design Applied to a Membrane Protein: Cyclooxygenase- 2, a Target for Arthritis.
et al: Anna M. Stevens, Jennifer L. Edwards, Roderick S. Stegeman, James K. Gierse, Carol M. Koboldt, William C. Stallings.

02:00 - 02:30 PM
Keith Watenpaugh. Invited Lecture.
Structure- Based Design of a Drug Effective Against a Changing Target.

02:30 - 03:00 PM
Ward Smith. Invited Lecture.
New Insights Into the Design of Inhibitors of Human Osteoclast Cathepsin K Based on the Structure of Inhibitor Complexes.

03:00 - 03:30 PM
Coffee Break.

03:30 - 04:00 PM WII02
(E465)
Jens J. Birktoft. Invited Lecture.
An IL-2: Peptidomimetic Complex as a Paradigm for Antagonizing Protein- Protein Interactions.
et al: C. Cook, R. Crowther, S. D. Emerson, D. C. Fry, U. Kammlott, R. Palermo, D. Weber, C.-M. Liu, Et Al.

04:00 - 04:30 PM
Panel Discussion.


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Last updated: Tue Jun 24 16:07:58 EDT 1997